The MolDarT is a novel short-term assay for testing mechanism-based molecular effects in developing zebrafish embryos. The objective of this study was to evaluate the inducibility of vitellogenin1 mRNA (Vtg1) by the estrogenically active compounds 17beta-Estradiol (E2), 17alpha-Ethinylestradiol (EE2), Nonylphenol (NP), Bisphenol A (BPA), Cyproconazol, and the suspected xeno-estrogen Atrazin in the MolDarT. Freshly fertilized zebrafish eggs were exposed semistatically for 120 h. Using reverse transcription real-time PCR, the relative abundance of Vtg1 was measured. For EE2 a dose-response relationship was established with EC50 = 60.7 ng/L (205 pM). Induction of Vtg1 was significant at concentrations of 84 pM EE2 (25 ng EE2/L) and above, 10 nM E2 (2.7 microg E2/L), 100 nM E2 (27 microg E2/L), 10 microM BPA (2280 microg BPA/L), and 15 microM BPA (3420 microg BPA/L). At NP concentrations of 0.75 microM (165 microg NP/L) and 1.5 microM (330 microg NP/L) Vtg1 was significantly down-regulated. Both atrazine and cyproconazol showed no effect on relative Vtg1 abundance. With this study we further characterize the MolDarT assay and show its applicability for effect screening of compounds.

译文

:MolDarT是一种新颖的短期测定法,用于测试斑马鱼胚胎发育中基于机理的分子效应。这项研究的目的是评估雌激素活性化合物17β-雌二醇(E2),17α-乙炔雌二醇(EE2),壬基酚(NP),双酚A(BPA),环丙唑醇和在MolDarT中疑似异种雌激素Atrazin。将新鲜受精的斑马鱼卵半静态暴露120 h。使用逆转录实时PCR,测量Vtg1的相对丰度。对于EE2,建立的剂量反应关系为EC50 = 60.7 ng / L(205 pM)。在84 pM EE2(25 ng EE2 / L)和更高浓度,10 nM E2(2.7 microg E2 / L),100 nM E2(27 microg E2 / L),10 microM BPA(2280 microg BPA)的浓度下,Vtg1的诱导作用显着/ L)和15 microM BPA(3420 microg BPA / L)。在0.75 microM(165 microg NP / L)和1.5 microM(330 microg NP / L)的NP浓度下,Vtg1显着下调。阿特拉津和环丙康唑均未显示相对Vtg1丰度的影响。通过这项研究,我们进一步表征了MolDarT分析并显示了其对化合物效果筛选的适用性。

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