Chemical biology is an emerging field that enables the study and manipulation of biological systems with probes whose reactivities provide structural insights. The opportunistic fungal pathogen Cryptococcus neoformans possesses a polysaccharide capsule that is a major virulence factor, but is challenging to study. We report here the synthesis of a hydroxylamine-armed fluorescent probe that reacts with reducing glycans and its application to study the architecture of the C. neoformans capsule under a variety of conditions. The probe signal localized intracellularly and at the cell wall-membrane interface, implying the presence of reducing-end glycans at this location where the capsule is attached to the cell body. In contrast, no fluorescence signal was detected in the capsule body. We observed vesicle-like structures containing the reducing-end probe, both intra- and extracellularly, consistent with the importance of vesicles in capsular assembly. Disrupting the capsule with DMSO, ultrasound, or mechanical shear stress resulted in capsule alterations that affected the binding of the probe, as reducing ends were exposed and cell membrane integrity was compromised. Unlike the polysaccharides in the assembled capsule, isolated exopolysaccharides contained reducing ends. The reactivity of the hydroxylamine-armed fluorescent probe suggests a model for capsule assembly whereby reducing ends localize to the cell wall surface, supporting previous findings suggesting that this is an initiation point for capsular assembly. We propose that chemical biology is a promising approach for studying the C. neoformans capsule and its associated polysaccharides to unravel their roles in fungal virulence.

译文

化学生物学是一个新兴领域,可以通过探针研究和操纵生物系统,探针的反应性提供了结构见解。机会性真菌病原体新型隐球菌具有多糖胶囊,是主要的毒力因子,但研究具有挑战性。我们在这里报告了与还原性聚糖反应的羟胺武装荧光探针的合成及其在各种条件下研究新孢子虫胶囊结构的应用。探针信号位于细胞内和细胞壁-膜界面处,这意味着在胶囊附着于细胞体的位置存在还原端聚糖。相反,在胶囊体内未检测到荧光信号。我们观察到在细胞内和细胞外均包含还原端探针的囊泡状结构,这与囊泡在荚膜组装中的重要性一致。用DMSO,超声或机械剪切应力破坏胶囊会导致胶囊改变,从而影响探针的结合,因为减少端暴露了,细胞膜的完整性受到损害。与组装胶囊中的多糖不同,分离的胞外多糖含有还原端。羟胺武装荧光探针的反应性表明了胶囊组装的模型,其中还原端定位于细胞壁表面,支持先前的发现,表明这是胶囊组装的起点。我们认为化学生物学是研究新生梭菌胶囊及其相关多糖以阐明其在真菌毒力中的作用的一种有前途的方法。

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