The preparation and stability parameters of para-acyl-calix[4]arene based solid lipid nanoparticles (SLNs) have been investigated. Atomic force microscopy (AFM) and photon correlation spectroscopy (PCS) show a mean particle size of 130 nm. In terms of preparation parameters, using the solvent displacement method, the nature and the volume of the organic solvent, the concentration of the amphiphile and the presence of a co-surfactant in the organic phase have been shown to affect significantly the size of the produced SLNs. In contrast, the stirring speed, the viscosity and the acidity of the aqueous phase and the amphiphile hydrophobic chain length have been shown to have no effect. In terms of stability parameters, the ionic strength has been shown to affect the short-time SLN stability depending on both the anion and the cation studied, with sodium sulphate causing precipitation. Ultrasonic, ultraviolet or microwave treatments of the SLN suspensions have no effect on the size of the SLNs. The study of the effects of short time thermal treatment revealed that the SLNs are not affected by one freezing-defreezing cycle and are stable at 100 degrees C in suspension. It is difficult to reconstitute the SLN suspensions after freeze-drying. Finally, the temporal stability of these suspensions in water has been shown to be superior to 1 year. The long-term temporal stability of suspensions stored in saline solution has been investigated. It has been demonstrated that the most destabilising effects arise from the presence in the storage suspension of sulphate ions.1H NMR, X-ray powder diffraction (XPD) and AFM have also been carried out on the calix-arene based SLNs and demonstrate the presence of a semi-organised matrix structure for the SLNs.

译文

:研究了对酰基杯[4]芳烃基固体脂质纳米颗粒(SLNs)的制备和稳定性参数。原子力显微镜(AFM)和光子相关光谱(PCS)显示平均粒径为130 nm。在制备参数方面,已证明使用溶剂置换法,有机溶剂的性质和体积,两亲物的浓度以及有机相中助表面活性剂的存在会显着影响产物的大小。 SLN。相反,已显示搅拌速度,水相的粘度和酸度以及两亲性疏水链长度没有影响。就稳定性参数而言,已证明离子强度会影响短期SLN稳定性,具体取决于所研究的阴离子和阳离子,而硫酸钠会引起沉淀。 SLN悬浮液的超声波,紫外线或微波处理对SLN的大小没有影响。对短时间热处理效果的研究表明,SLN不受一个冷冻-解冻循环的影响,并且在100℃的悬浮状态下稳定。冷冻干燥后很难重新配制SLN悬浮液。最后,这些悬浮液在水中的时间稳定性已证明优于1年。已经研究了盐溶液中储存的悬浮液的长期时间稳定性。业已证明,最不稳定的作用是由硫酸根离子的储存悬浮液引起的。1HNMR,X射线粉末衍射(XPD)和AFM也在基于芳烃芳烃的SLN上进行,并证明了存在SLN的半组织矩阵结构。

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