Surface potential difference, conductance, and elasticity changes of bilayer lipid membranes induced by the antivirus drugs amantadine and remantadine were measured. An influence on the human erythrocyte shape was shown. Both drugs are stomatocytogenic. The adsorption at the cytoplasmatic membrane was electrophoretically proved. The heat-induced vesiculation is partly inhibited. No microvesicles were observed. Instead, large tails which did not detach from the cell body were seen. The general conclusion is that these amphiphilic adamantane derivatives are membrane agents which modify membrane interaction processes, possibly by influencing the bending properties.

译文

测量了抗病毒药物金刚烷胺和remantadine引起的双层脂质膜的表面电位差,电导和弹性变化。显示了对人红细胞形状的影响。两种药物都是造口剂。电泳证明了在细胞质膜上的吸附。热诱导的囊泡被部分抑制。未观察到微泡。相反,看到了没有从细胞体上脱离的大尾巴。一般结论是,这些两亲性金刚烷衍生物是膜剂,可能通过影响弯曲性能来改变膜相互作用过程。

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