The incretin - glucose-dependent insulinotropic polypeptide (GIP) - and the pro-inflammatory cytokine osteopontin are known to have important roles in the regulation of adipose tissue functions. In this work we show that GIP stimulates lipogenesis and osteopontin expression in primary adipocytes. The GIP-induced increase in osteopontin expression was inhibited by the NFAT (the transcription factor nuclear factor of activated T-cells) inhibitor A-285222. Also, the NFAT kinase glycogen synthase kinase (GSK) 3 was upregulated by GIP. To test whether cAMP might be involved in GIP-mediated effects on osteopontin a number of strategies were used. Thus, the β3-adrenergic receptor agonist CL316,243 stimulated osteopontin expression, an effects which was mimicked by OPC3911, a specific inhibitor of phosphodiesterase 3. Furthermore, treatment of phosphodiesterase 3B knock-out mice with CL316,243 resulted in a dramatic upregulation of osteopontin in adipose tissue which was not the case in wild-type mice. In summary, we delineate mechanisms by which GIP stimulates osteopontin in adipocytes. Given the established link between osteopontin and insulin resistance, our data suggest that GIP by stimulating osteopontin expression, also could promote insulin resistance in adipocytes.

译文

已知肠促胰岛素素-葡萄糖依赖性促胰岛素多肽 (GIP) -和促炎细胞因子骨桥蛋白在调节脂肪组织功能中起重要作用。在这项工作中,我们表明GIP刺激原代脂肪细胞中的脂肪生成和骨桥蛋白表达。GIP诱导的骨桥蛋白表达的增加被NFAT (活化T细胞的转录因子核因子) 抑制剂A-285222抑制。此外,GIP上调了NFAT激酶糖原合酶激酶 (GSK) 3。为了测试cAMP是否可能参与GIP介导的对骨桥蛋白的作用,使用了许多策略。因此,β3-肾上腺素能受体激动剂CL316 243刺激骨桥蛋白表达,这种作用被磷酸二酯酶3的特异性抑制剂OPC3911模仿。此外,用CL316 243处理磷酸二酯酶3B敲除小鼠导致脂肪组织中骨桥蛋白的显著上调,这在野生型小鼠中并非如此。总之,我们描述了GIP刺激脂肪细胞中的骨桥蛋白的机制。鉴于已建立的骨桥蛋白与胰岛素抵抗之间的联系,我们的数据表明GIP通过刺激骨桥蛋白的表达也可以促进脂肪细胞的胰岛素抵抗。

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