Cationic antimicrobial peptides are produced by almost all species of life as a component of their immediate non-specific defense against infections. The assets of these peptides in clinical application include their potential for broad-spectrum activity, rapid bactericidal activity and low propensity for resistance development, whereas possible disadvantages include their high cost, limited stability (especially when composed of L-amino acids), and unknown toxicology and pharmacokinetics. Initial barriers to their success are being increasingly overcome with the development of stable, more cost-effective and potent broad-spectrum synthetic peptides. Thus, there is hope that they will spawn a new generation of antimicrobials with a broad range of topical and systemic applications against infections.

译文

:阳离子抗菌肽几乎是生活中所有物种所产生的,它们是针对感染的直接非特异性防御​​的组成部分。这些肽在临床应用中的资产包括它们具有广谱活性,快速杀菌活性和耐药性发展倾向的潜力,而可能的缺点包括它们的成本高,稳定性有限(尤其是由L-氨基酸组成时)和未知的毒理学和药代动力学。随着稳定,更具成本效益和有效的广谱合成肽的开发,克服其成功的最初障碍越来越多。因此,希望它们能够产生新一代的抗菌药,具有广泛的局部和全身应用来抵抗感染。

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