The nitroxyl (HNO) donor Angeli's salt (Na(2)N(2)O(3); AS) is cytotoxic in vitro, inducing double strand DNA breaks and base oxidation, yet may have pharmacological application in the treatment of cardiovascular disease. The chemical profiles of AS and synthetic peroxynitrite (ONOO(-)) in aerobic solution were recently compared, and AS was found to form a distinct reactive intermediate. However, similarities in the chemical behavior of the reactive nitrogen oxide species (RNOS) were apparent under certain conditions. Buffer composition was found to have a significant and unexpected impact on the observed chemistry of RNOS, and varied buffer conditions were utilized to further distinguish the chemical profiles elicited by the RNOS donors AS and synthetic ONOO(-). Addition of HEPES to the assay buffer significantly quenched oxidation of dihydrorhodamine (DHR), hydroxylation of benzoic acid (BA), and DNA damage by both AS and ONOO(-), and oxidation and nitration of hydroxyphenylacetic acid by ONOO(-). Additionally, H(2)O(2) was produced in a concentration-dependent manner from the interaction of HEPES with both the donor intermediates. Interestingly, clonogenic survival was not affected by HEPES, indicating that H(2)O(2) is not a contributing factor to in vitro cytotoxicity of AS. Variation in RNOS reactivity was dramatic with significantly higher relative affinity for the AS intermediate toward DHR, BA, DNA, and HEPES and increased production of H(2)O(2). Further, AS reacted to a significantly greater extent with the unprotonated amine form of HEPES while the interaction of ONOO(-) with HEPES was pH-independent. Addition of bicarbonate only altered ONOO(-) chemistry. This study emphasizes the importance of buffer composition on chemical outcome and thus on interpretation and provides further evidence that ONOO(-) is not an intermediate formed between the reaction of O(2) and HNO produced by AS.

译文

硝基 (HNO) 供体Angeli盐 (Na(2)N(2)O(3); AS) 在体外具有细胞毒性,可诱导双链DNA断裂和碱基氧化,但可能在治疗心血管疾病中具有药理应用。最近比较了好氧溶液中AS和合成过氧亚硝酸盐 (ONOO(-)) 的化学特征,发现AS形成了独特的反应性中间体。然而,在某些条件下,反应性氮氧化物物种 (RNOS) 的化学行为相似。发现缓冲液成分对观察到的RNOS化学有重大且出乎意料的影响,并且利用不同的缓冲液条件来进一步区分RNOS供体AS和合成ONOO(-) 引起的化学特征。将HEPES添加到测定缓冲液中可以显着淬灭二氢罗丹明 (DHR) 的氧化,苯甲酸 (BA) 的羟基化以及AS和ONOO(-) 的DNA损伤,以及ONOO(-) 的羟基苯乙酸的氧化和硝化。此外,由HEPES与两种供体中间体的相互作用以浓度依赖性方式产生H(2)O(2)。有趣的是,克隆形成的存活不受HEPES的影响,表明H(2)O(2) 不是AS体外细胞毒性的影响因素。RNOS反应性的变化非常明显,AS中间体对DHR,BA,DNA和HEPES的相对亲和力明显更高,H(2)O(2) 的产生增加。此外,AS与HEPES的未质子化胺形式的反应程度明显更高,而ONOO(-) 与HEPES的相互作用与pH无关。添加碳酸氢盐只会改变ONOO(-) 化学性质。这项研究强调了缓冲液组成对化学结果以及解释的重要性,并提供了进一步的证据,表明ONOO(-) 不是O(2) 和AS产生的HNO反应之间形成的中间体。

+1
+2
100研值 100研值 ¥99课程
检索文献一次
下载文献一次

去下载>

成功解锁2个技能,为你点赞

《SCI写作十大必备语法》
解决你的SCI语法难题!

技能熟练度+1

视频课《玩转文献检索》
让你成为检索达人!

恭喜完成新手挑战

手机微信扫一扫,添加好友领取

免费领《Endnote文献管理工具+教程》

微信扫码, 免费领取

手机登录

获取验证码
登录